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Adrenergic Pharmacology
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Revision as of 06:16, 4 February 2023
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06:16, 4 February 2023
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Line 24:
*↓insulin release, ↓lipolysis, ↓aqueous humor production
*↓insulin release, ↓lipolysis, ↓aqueous humor production
|
|
−
presynaptic G<sub>i</sub> → ↓AC → ↓cAMP → ↓NT release
, sympatholytic effects
+
presynaptic G<sub>i</sub> → ↓AC → ↓cAMP → ↓NT release
|
|
*Dexmedetomidine
*Dexmedetomidine
Line 59:
Line 59:
*↑aqueous humor production
*↑aqueous humor production
|
|
−
G<sub>s</sub> → ↑cAMP → ↑PKA
+
G<sub>s</sub>
→ ↑AC;
→ ↑cAMP → ↑PKA
|
|
*Albuterol
*Albuterol
Line 76:
Line 76:
*Labet'''alol''' (anti-α1)
*Labet'''alol''' (anti-α1)
|-
|-
−
| β3 || Iso > Epi = NE
||
Lipolysis
, bladder
detrusor relaxation |
| Gs,
cAMP
up
+
| β3 || Iso > Epi = NE
+
*
Lipolysis
+
*Bladder
detrusor relaxation
+
|
+
G<sub>s</sub> → ↑AC; → ↑
cAMP
→ ↑PKA
|
|
*Mirabegron
*Mirabegron
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